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INDOLE DERIVATIVES AND PROCESS FOR THEIR PREPARATI

来源:东饰资讯网
专利内容由知识产权出版社提供

专利名称:INDOLE DERIVATIVES AND PROCESS FOR

THEIR PREPARATION

发明人:ABEL, Ulrich申请号:EP11779145.9申请日:20111027公开号:EP2632897A1公开日:20130904

摘要:Substituted indole derivatives of formula (I) wherein the radicals have e. g. thefollowing meaning: R is hydrogen, -C-alkyl, R is hydrogen, -C-alkyl or cycloC-alkyl; R is ORR is hydrogen or halogen, R is hydrogen, -C-alkyl R is hydrogen, -C-alkyl R is hydrogen or-C-alkyl; X is a group -C(O)CH- or -CH=CH-; R is hydrogen are potent inhibitors of Abetapeptide polymerization and can be used for the treatment of e.g. Alzheimers disease orocular disorders.

申请人:Merz Pharma GmbH & Co. KGaA

地址:Eckenheimer Landstrasse 100 60318 Frankfurt am Main DE

国籍:DE

代理机构:Jacobi, Markus Alexander

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